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Cyclobenzaprine HCl 1%/Diclofenac Sodium 1%/Gabapentin 3%/Ibuprofen 10%/Tetracaine 2% Topical Gel

This formulation is a combination of Cyclobenzaprine HCl 1%, Diclofenac Sodium 1%, Gabapentin 3%, Ibuprofen 10%, and Tetracaine 2% in a topical gel. It is a semisolid formulation dispensed through a pump mechanism, which allows for easy and precise application on the skin. The gel-like consistency ensures targeted treatment or absorption of the active ingredients.

The formulation is designed to treat a variety of disease states. Cyclobenzaprine HCl is a muscle relaxant used to relieve muscle spasms, Diclofenac Sodium is a nonsteroidal anti-inflammatory drug (NSAID) used to treat pain and inflammation, Gabapentin is used to manage nerve pain, Ibuprofen is another NSAID used to reduce pain, inflammation, and fever, and Tetracaine is a local anesthetic used to numb the skin. The combination of these ingredients provides comprehensive pain management and relief from inflammation.

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Topical Gel
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Formula Information

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This formulation is a unique combination of five active ingredients: Cyclobenzaprine HCl 1%, Diclofenac Sodium 1%, Gabapentin 3%, Ibuprofen 10%, and Tetracaine 2%. Each of these ingredients plays a crucial role in managing various disease states. The formulation is designed as a semisolid gel, which is dispensed through a pump mechanism. This design allows for easy and precise application on the skin, ensuring targeted treatment and optimal absorption of the active ingredients.

Cyclobenzaprine HCl is a muscle relaxant that works by blocking nerve impulses (or pain sensations) that are sent to your brain. It is commonly used to treat muscle spasms and to relieve pain, stiffness, and discomfort caused by strains, sprains, or injuries to your muscles. Diclofenac Sodium is a nonsteroidal anti-inflammatory drug (NSAID) that reduces substances in the body that cause pain and inflammation. It is used to treat mild to moderate pain, or signs and symptoms of osteoarthritis or rheumatoid arthritis.

Gabapentin is an anticonvulsant that is often used to relieve nerve pain following shingles (a painful rash due to herpes zoster infection) in adults. It is also used to treat neuropathic pain, a type of long-lasting pain caused by damage to the nerves. Ibuprofen is another NSAID that works by reducing hormones that cause inflammation and pain in the body. It is used to reduce fever and treat pain or inflammation caused by many conditions such as headache, toothache, back pain, arthritis, menstrual cramps, or minor injury. Tetracaine is a local anesthetic that is used to numb different parts of the body before certain medical procedures or to relieve the pain, itching, or discomfort caused by certain skin conditions.

This formulation, therefore, provides a comprehensive approach to pain management, addressing not only the symptoms but also the underlying causes of pain. It is particularly useful for patients suffering from conditions that cause chronic or acute pain, such as arthritis, nerve damage, muscle spasms, and certain skin conditions. The gel-like consistency and the pump mechanism allow for easy application and precise dosing, ensuring that the medication is delivered exactly where it is needed.

If you have any questions about this formulation, its uses, or how it can benefit you or your patients, please do not hesitate to reach out to us. Our team of knowledgeable compounding pharmacists at Bayview Pharmacy is always here to help.

Drug Interactions

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This formulation contains a combination of Cyclobenzaprine HCl, Diclofenac Sodium, Gabapentin, Ibuprofen, and Tetracaine. These active ingredients work together to provide relief from pain and inflammation associated with various conditions such as arthritis, nerve pain, muscle spasms, and other similar conditions. However, it's important to be aware of potential drug interactions that may occur with this formulation.

Cyclobenzaprine HCl, a muscle relaxant, may interact with drugs like monoamine oxidase inhibitors (MAOIs), certain antidepressants, and alcohol, leading to increased sedation and potentially serious health risks. Diclofenac Sodium, a nonsteroidal anti-inflammatory drug (NSAID), may interact with blood thinners, blood pressure medications, and other NSAIDs, potentially increasing the risk of bleeding or kidney problems. It's also important to avoid alcohol while using this medication as it can increase the risk of stomach bleeding.

Gabapentin, used to treat nerve pain, may interact with antacids, morphine, and hydrocodone, potentially affecting the way these drugs work. It's also important to avoid alcohol while using this medication as it can increase the risk of side effects. Ibuprofen, another NSAID in this formulation, may interact with blood thinners, blood pressure medications, and other NSAIDs, potentially increasing the risk of bleeding or kidney problems. It's also important to avoid alcohol while using this medication as it can increase the risk of stomach bleeding.

Tetracaine, a local anesthetic, has fewer interactions but may interact with certain heart medications and other local anesthetics. It's also important to avoid applying this medication to broken or inflamed skin as it can increase the risk of side effects.

It's crucial to inform your healthcare provider about all the medications you're currently taking, including prescription drugs, over-the-counter medications, vitamins, and herbal supplements, to avoid potential drug interactions. If you're pregnant, planning to become pregnant, or breastfeeding, discuss with your healthcare provider before using this formulation as certain ingredients may pose risks to the baby.

Always use this medication as directed by your healthcare provider. Do not use more than the recommended dose or for longer than prescribed. If you experience any side effects or if your condition does not improve or worsens, contact your healthcare provider immediately.

If you have any questions or concerns about this formulation, please do not hesitate to reach out to us. We are here to help and provide you with the most accurate and up-to-date information.

How Does it Work

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This formulation is a combination of five active ingredients: Cyclobenzaprine HCl, Diclofenac Sodium, Gabapentin, Ibuprofen, and Tetracaine, each with a unique mechanism of action that contributes to the overall therapeutic effect of the gel.

Cyclobenzaprine HCl is a muscle relaxant that works by blocking nerve impulses (or pain sensations) that are sent to your brain. It is particularly effective in treating muscle spasms and associated pain. Diclofenac Sodium is a nonsteroidal anti-inflammatory drug (NSAID) that reduces substances in the body that cause pain and inflammation. It is commonly used to treat mild to moderate pain, or signs and symptoms of osteoarthritis or rheumatoid arthritis.

Gabapentin is an anticonvulsant and nerve pain medication. It works by calming down nerve activity to reduce pain sensations. It is often used to treat nerve pain caused by shingles (postherpetic neuralgia) or other nerve pain conditions. Ibuprofen is another NSAID that works by reducing hormones that cause inflammation and pain in the body. It is used to reduce fever and treat pain or inflammation caused by many conditions such as headache, toothache, back pain, arthritis, menstrual cramps, or minor injury.

Tetracaine is a local anesthetic that works by blocking nerve signals in your body. It is used to numb different parts of the body before medical procedures or to relieve pain and itching caused by certain skin conditions. When applied topically, Tetracaine can help to numb the skin and surrounding area, providing relief from pain and discomfort.

When these five active ingredients are combined in a gel formulation, they work together to provide targeted relief from pain and inflammation. The gel is designed to be easily applied to the skin, allowing for the active ingredients to be absorbed directly into the affected area. This targeted approach can provide faster and more effective relief compared to oral medications, as it bypasses the digestive system and goes straight to the source of the pain.

If you have any questions about this formulation or how it works, please don't hesitate to reach out to us at Bayview Pharmacy. Our team of knowledgeable compounding pharmacists is always here to help.

Other Uses

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This multi-drug combination topical gel formulation contains numerous active components, each with its own distinct therapeutic properties. While its primary usage is for localized analgesic and anti-inflammatory effects, it can also be employed in a wider range of conditions. Other possible uses range from the management of symptoms in conditions such as osteoarthritis, fibromyalgia, and diabetic peripheral neuropathy, where it can be utilized to manage chronic pain, inflammation, and neuropathic pain symptoms effectively, given its anti-inflammatory and analgesic constituents.

Furthermore, the inclusion of Tetracaine, a local anesthetic, could have potential use in surface anesthesia for minor surgical procedures, including skin grafts or minor plastic surgery procedures when systemic anesthesia is not required. Its action could also be beneficial in post-herpetic neuralgia, a chronic pain symptom following an outbreak of shingles. The inclusion of Cyclobenzaprine HCl, a muscle relaxant, indicates that this formulation could also be useful in alleviating muscle spasms and associated pain, providing more comprehensive pain management."

However, as the formulation includes multiple active components, rapid escalation in conditions or pain levels should be monitored closely as this could indicate a need for a revised approach to treatment. Always consult your healthcare provider for appropriate management and prescription.

Please note that although the medicine has potential therapeutic benefits in these conditions, it is not a substitute for systematic therapy or a comprehensive care plan. It is crucial that it should be used as a part of an overall management plan under the supervision of a healthcare provider. Patients should possess an understanding of how to correctly administer a topical gel, including the appropriate area, quantity, and frequency of application.

If there are any further queries or concerns about the various uses of this compound or dosage form, feel free to reach out to our knowledge team at Bayview Pharmacy. Our aim is to provide personalized and detailed information that will foster understanding and promote proper use of our products and services.

Frequently Asked Questions

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What is the use of this compounded formulation?

This compounded formulation contains Cyclobenzaprine HCl, Diclofenac Sodium, Gabapentin, Ibuprofen and Tetracaine. It's used topically on the skin to help treat pain, inflammation, muscle spasms and nerve disorders.

How do I apply this medication?

You apply this medicine topically on the skin, using the pump mechanism to dispense the correct dosage. Apply it as prescribed your healthcare provider.

How often should I use this gel?

Usage depends on your doctor's recommendation, your treatment needs, and your skin's response to the medication. Do not use more or less often than directed.

What happens if I miss a dose?

If you miss a dose, apply it as soon as you remember. If it's close to your next dosage time, skip the missed dose and stick to the regular schedule.

Are there any side effects to this medication?

Side effects can include skin irritation or sensitivity. If you experience any unusual side effects or reactions, such as rashes, itching, or swelling, contact your healthcare provider immediately.

Can this gel be used with other topical medications?

Do not use this gel with other topical medications unless directed by your healthcare provider, as it could cause drug interactions.

Should I cover the applied area with a bandage after using the gel?

Unless your healthcare provider advises you to, do not cover the area where you have applied the gel. It's designed to be absorbed directly through the skin.

Should I rub the gel completely into my skin?

Yes, gently rub the gel into your skin for maximum absorption. However, you should not rub it in so hard that it causes irritation or discomfort.

Can I apply this gel on open wounds or damaged skin?

No, avoid applying this formulation on open wounds, cuts, burns, or damaged skin unless instructed by your healthcare provider.

Do I need to wash my hands after applying this gel?

Yes, you should wash your hands thoroughly after applying this medication to avoid accidental contact with your eyes or mouth, unless your hands are the area of treatment.

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Formulas and/or material listed are not to be interpreted as a promise, guarantee or claim of therapeutic efficacy or safety. The information contained herein is not intended to replace or substitute for conventional medical care, or encourage its abandonment. Every patient is unique, and formulas should be adjusted to meet their individual needs.

No compounded medications are reviewed by the FDA for safety or efficacy.