Sublingual Semaglutide (generic Ozempic®) now available! Get Started
Dashboard
Formulas

Cyclobenzaprine 0.5%/Ketoprofen 5% Topical Gel

This formulation combines Cyclobenzaprine 0.5% and Ketoprofen 5% in a topical gel. Cyclobenzaprine is a muscle relaxant that works by blocking nerve impulses (or pain sensations) that are sent to your brain. Ketoprofen is a nonsteroidal anti-inflammatory drug (NSAID) that reduces hormones that cause inflammation and pain in the body. Together, they provide targeted treatment for conditions such as muscle spasms, inflammation, and pain.

The gel is a semisolid formulation dispensed through a pump mechanism, which allows for easy and precise application on the skin. This facilitates the absorption of the active ingredients directly at the site of discomfort, providing localized relief. The gel-like consistency ensures a smooth application without causing any discomfort or residue on the skin.

Want a different strength?
Click the Text Us button below.
To prescribe, you must be a verified prescriber.
To prescribe, you must be in a state where we hold an active out-of-state pharmacy license.
Starting at
Must be E-Prescribed
Get Started
Generate LeafletShow Leaflet
This medication requires a prescription from your doctor
Trusted by 60,357 patients to date.
A group of faces of our past satisfied patients.
A svg symbol of a mortar and pestle with ingredients going in.
Custom made in our compounding labs.
Sliders that show the customization of ingredients.
Personalized treatment for better results.
User with a gear showing the personalization of the formulation.
All strengths and ingredients are tailored to your needs.
This medication is not available at retail pharmacies. It is compounded, and may be more effective at treating you or your patient.
Ketoprofen
Cyclobenzaprine Hydrochloride
Topical Gel
653f482be23ed933a97647b2
Thank you! Your submission has been received!
Oops! Something went wrong while submitting the form.
Loading icon rotating.
Thank you! Your submission has been received!
Oops! Something went wrong while submitting the form.

Dosing Calculator

Get general dosing information for a patient by using this calculator.
Thank you! Your submission has been received!
Oops! Something went wrong while submitting the form.
Loading icon rotating.
Thank you! Your submission has been received!
Oops! Something went wrong while submitting the form.

Formula Information

A small arrow pointing down

This formulation combines two active ingredients, Cyclobenzaprine and Ketoprofen, in a topical gel format. Cyclobenzaprine is a muscle relaxant that works by blocking nerve impulses (or pain sensations) that are sent to your brain. Ketoprofen is a nonsteroidal anti-inflammatory drug (NSAID) that reduces hormones that cause inflammation and pain in the body. The combination of these two ingredients provides both pain relief and muscle relaxation.

The gel is a semisolid formulation that is dispensed through a pump mechanism. This allows for easy and precise application on the skin. The gel-like consistency ensures that the active ingredients are absorbed effectively into the skin for targeted treatment. This is particularly beneficial for localized pain and inflammation, as the medication can be applied directly to the affected area.

This formulation is used to treat a variety of disease states. Cyclobenzaprine is often used to treat muscle spasms caused by painful muscle conditions. It is usually used along with rest and physical therapy. Ketoprofen is used to relieve pain, swelling, and joint stiffness caused by arthritis. This medication is also used to treat mild to moderate pain, and to reduce fever. The combination of these two medications in a topical gel format allows for targeted treatment of these conditions.

It is important to use this medication as directed by your healthcare provider. The amount of gel needed will depend on the size of the area to be treated. The gel should be applied to the affected area and rubbed in gently until it is absorbed. Avoid applying this medication to broken skin or open wounds. Also, this medication should not be used in the eyes, nose, or mouth. If you have any questions about how to use this medication, please reach out to us.

As with any medication, there may be potential side effects. These can include skin irritation at the application site, dizziness, dry mouth, or constipation. If any of these side effects persist or worsen, contact your healthcare provider immediately. It is also important to inform your healthcare provider of all the medications you are currently taking, as there may be potential interactions with this topical gel.

Overall, this Cyclobenzaprine 0.5%/Ketoprofen 5% Topical Gel is an effective treatment option for pain and inflammation. It provides targeted treatment with the convenience of a topical application. If you have any questions or concerns about this formulation, please do not hesitate to reach out to us at Bayview Pharmacy. We are a team of knowledgeable compounding pharmacists, and we are here to help.

Drug Interactions

A small arrow pointing down

The combination of Cyclobenzaprine and Ketoprofen in a topical gel formulation is primarily used for the management of localized pain and inflammation. Cyclobenzaprine, a muscle relaxant, works by blocking nerve impulses (or pain sensations) that are sent to your brain. Ketoprofen, on the other hand, is a nonsteroidal anti-inflammatory drug (NSAID) that reduces hormones that cause inflammation and pain in the body.

While this formulation is generally considered safe for most patients, it's important to be aware of potential drug interactions. Cyclobenzaprine may interact with other medications that cause drowsiness such as opioid pain or cough relievers, alcohol, marijuana, drugs for sleep or anxiety, other muscle relaxants, or antihistamines. Additionally, some medications can affect the removal of cyclobenzaprine from your body, which may affect how cyclobenzaprine works. Examples include certain anti-seizure drugs, cimetidine, and certain antidepressants.

Ketoprofen may interact with other NSAIDs, increasing the risk of stomach ulcers and bleeding. It can also interact with blood thinners, corticosteroids, and certain medications for high blood pressure. If you are taking aspirin to prevent heart attack or stroke, ketoprofen can make aspirin less effective in protecting your heart and blood vessels. If you are taking any of these medications, it's important to discuss this with your healthcare provider.

It's also important to note that this formulation should not be used with other topical products, including sunscreens, lotions, or cosmetics, as this may alter the absorption of the active ingredients. Additionally, avoid exposure to heat, as this can increase the absorption of the medication, potentially leading to increased side effects.

As with any medication, it's important to use this formulation as directed by your healthcare provider. If you have any questions or concerns about potential drug interactions or how to use this medication, please don't hesitate to reach out to us at Bayview Pharmacy. We're here to help ensure that you receive the most benefit from your medications.

How Does it Work

A small arrow pointing down

The Cyclobenzaprine 0.5%/Ketoprofen 5% Topical Gel is a unique formulation that combines the muscle relaxant properties of Cyclobenzaprine and the anti-inflammatory effects of Ketoprofen. This combination is designed to provide targeted relief from pain and inflammation associated with various musculoskeletal conditions.

Cyclobenzaprine, the first active ingredient, is a muscle relaxant that works by blocking nerve impulses (or pain sensations) that are sent to your brain. It is particularly effective in treating muscle spasms and associated pain. When applied topically, Cyclobenzaprine acts locally on the affected area, reducing muscle tension and providing relief from discomfort.

Ketoprofen, the second active ingredient, is a nonsteroidal anti-inflammatory drug (NSAID). It works by reducing hormones that cause inflammation and pain in the body. When applied topically, Ketoprofen can directly target the site of inflammation, reducing swelling and pain without the systemic side effects often associated with oral NSAIDs.

The gel formulation allows for easy application and absorption of the active ingredients. The semisolid consistency of the gel ensures that the medication stays on the skin longer, allowing for better absorption and more effective treatment. The pump mechanism of the container allows for precise dosing and application, ensuring that the patient receives the correct amount of medication every time.

This formulation is particularly effective in treating conditions such as arthritis, bursitis, and acute muscle or joint injuries. By reducing inflammation and relaxing the muscles, it can significantly improve mobility and quality of life for patients suffering from these conditions.

As with any medication, it is important to use this product as directed by a healthcare professional. Patients should apply the gel to the affected area as directed, and avoid contact with eyes, mouth, and other sensitive areas. If any adverse reactions occur, such as rash, itching, or difficulty breathing, contact a healthcare professional immediately.

If you have any questions about the Cyclobenzaprine 0.5%/Ketoprofen 5% Topical Gel, or if you would like more information about how it works, please don't hesitate to reach out to us at Bayview Pharmacy. Our team of knowledgeable compounding pharmacists is always here to help.

Other Uses

A small arrow pointing down

Cyclobenzaprine 0.5%/Ketoprofen 5% topical gel, in addition to its primary use for pain management, inflammation and muscle relaxation, can serve several other purposes. This unique compound formulation can be used off-label for various conditions related to pain and inflammation beyond those conditions for which it has been primarily indicated.

For instances, it has been employed by practitioners to manage different forms of arthritis, such as rheumatoid arthritis and osteoarthritis, due to its powerful analgesic and anti-inflammatory effects. Increasing evidence also suggests that it can be used in treating symptoms related to fibromyalgia, particularly in managing muscle stiffness and tenderness associated with this condition. Furthermore, it has been noted by some clinicians to lessen the pain associated with certain neuropathic conditions, given its nerve pain relieving properties.

Additionally, as a topical formulation, it minimizes the systemic absorption and therefore reduces the risk of potential adverse effects compared to oral dosage forms. This makes it an attractive alternative for patients who may be intolerant or unresponsive to traditional oral therapies. It can also be beneficial to patients who have difficulty swallowing tablets or capsules.

Finally, its semisolid form that can be easily dispensed through a pump mechanism makes it user-friendly and facilitates more accurate dosing. The targeted application benefits both the patient, by providing localized relief, and the prescriber, by tailoring treatment to the specific area of concern.

Before suggesting or using Cyclobenzaprine 0.5%/Ketoprofen 5% topical gel for any off-label indications, it's crucial to keep in mind that the efficacy of its use for non-indicated conditions may vary between patients and treatment should always be provided under the guidance and supervision of experienced healthcare providers. If you have any questions related to the use of this formulation, don't hesitate to reach out to us. Our team at Bayview Pharmacy is well equipped to provide appropriate counsel and support in your therapeutic choices.

Frequently Asked Questions

A small arrow pointing down

What is Cyclobenzaprine 0.5%/Ketoprofen 5% Topical Gel?

Cyclobenzaprine 0.5%/Ketoprofen 5% Topical Gel is a semisolid formulation that combines two active ingredients: Cyclobenzaprine and Ketoprofen. It is typically applied to the skin for targeted treatment and absorption.

How is the Cyclobenzaprine 0.5%/Ketoprofen 5% Topical Gel administered?

This topical gel is dispensed through a pump mechanism, which facilitates easy and precise application on the skin.

Can this topical gel be used for any skin type?

If you have a specific skin type or condition, it is recommended to discuss this with your healthcare provider before using this topical gel to ensure it is suitable for your skin.

What is the function of Cyclobenzaprine and Ketoprofen in the topical gel?

Cyclobenzaprine is a muscle relaxant that works by blocking nerve impulses (or pain sensations) that are sent to your brain. Ketoprofen is a nonsteroidal anti-inflammatory drug (NSAID) that works by reducing hormones that cause inflammation and pain in the body.

Is it safe to apply this gel on broken or irritated skin?

This topical gel should only be applied on intact or unbroken skin. Applying this product to open wounds or irritated skin may lead to unwanted side effects. Consult with your healthcare provider if you're unsure.

What should I do if I miss a dose?

Apply the missed dose as soon as you remember. However, if it is near the time of the next dose, skip the missed dose and resume your usual dosing schedule. Do not double the dose to catch up.

How should I store this topical gel?

Store this medication at room temperature, away from light and moisture. Do not store in the bathroom. Keep all medications away from children and pets.

Can I use other skin products while using this topical gel?

Before using other topical products, consult with your healthcare provider. There may be potential interactions or side effects if used with other skin products.

What happens if the gel accidentally gets into my eyes?

If the gel accidentally gets into your eyes, rinse thoroughly with water. Seek medical attention if you experience any discomfort or pain.

Can I use this topical gel if I'm pregnant or breastfeeding?

If you are pregnant or breastfeeding, it is important to consult with your healthcare provider before using this topical gel. The active ingredients may have potential effects on the baby.

Related Formulas

Related Products
Formulas and/or material listed are not to be interpreted as a promise, guarantee or claim of therapeutic efficacy or safety. The information contained herein is not intended to replace or substitute for conventional medical care, or encourage its abandonment. Every patient is unique, and formulas should be adjusted to meet their individual needs.

No compounded medications are reviewed by the FDA for safety or efficacy.