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Amitriptyline HCl 1%/Tetracaine HCl 2% Vaginal Cream

This formulation is a semisolid cream containing Amitriptyline HCl at a concentration of 1% and Tetracaine HCl at a concentration of 2%. It is dispensed in a tube for easy and accurate application in the vaginal area. The cream is specifically designed to deliver medication and provide therapeutic effects for certain gynecological conditions.

Amitriptyline HCl is a tricyclic antidepressant that is used off-label for pain management, while Tetracaine HCl is a local anesthetic. Together, they work synergistically to alleviate pain and discomfort associated with various gynecological conditions. This formulation is particularly beneficial for patients suffering from vulvodynia, a chronic pain condition in the vulvar area, and vestibulodynia, a subset of vulvodynia that is characterized by severe pain in the vestibule area of the vagina. It may also be used to manage pain associated with interstitial cystitis, a chronic condition causing bladder pressure and pain.

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Amitriptyline Hydrochloride
Tetracaine Hydrochloride
Vaginal Cream
65316cc373096c6cf9ae5370
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Formula Information

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This formulation is a compounded medication that combines Amitriptyline HCl at a concentration of 1% and Tetracaine HCl at a concentration of 2% in a vaginal cream. Amitriptyline HCl is a tricyclic antidepressant that has been found to be effective in managing chronic pain, while Tetracaine HCl is a potent local anesthetic. When combined in a cream formulation, these two active ingredients work synergistically to provide both pain relief and local anesthesia in the vaginal area.

The cream is a semisolid formulation that is dispensed in a tube for convenient and precise application. It is designed to deliver medication directly to the vaginal area, providing therapeutic effects for specific gynecological conditions. This targeted delivery system allows for the active ingredients to be absorbed directly into the affected area, providing faster relief and minimizing systemic side effects.

This formulation is commonly used to manage pain and discomfort associated with conditions such as vulvodynia, vestibulodynia, and other gynecological conditions that cause chronic pain. Amitriptyline HCl works by increasing the levels of certain chemicals in the brain that help improve the mood and reduce the sensation of pain. Tetracaine HCl, on the other hand, works by blocking nerve signals in the body, providing a numbing effect to the area where the cream is applied.

It is important to note that this medication should be used as directed by a healthcare provider. The cream should be applied to the affected area as directed, usually once or twice daily. It is not intended for oral, ophthalmic, or intravaginal use. Patients should wash their hands before and after applying the cream. If any side effects occur, such as irritation or an allergic reaction, patients should discontinue use and contact their healthcare provider immediately.

As with any medication, it is important to discuss any other medications, supplements, or health conditions with your healthcare provider before starting this treatment. This will help ensure that the medication is safe and effective for you.

If you have any questions about this formulation, please do not hesitate to reach out to us at Bayview Pharmacy. Our team of knowledgeable compounding pharmacists is here to help you understand your medication and how it can help manage your condition.

Drug Interactions

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Amitriptyline HCl and Tetracaine HCl are both active ingredients in this vaginal cream formulation. Amitriptyline is a tricyclic antidepressant that has analgesic properties, making it useful for pain management in certain gynecological conditions. Tetracaine is a local anesthetic that provides temporary numbness or loss of sensation in the area where it is applied, offering immediate relief from discomfort or pain.

It's important to be aware of potential drug interactions when using this formulation. Amitriptyline can interact with a number of medications, including MAO inhibitors, SSRIs, anticholinergic drugs, and certain antihypertensive drugs. Combining these medications can increase the risk of side effects such as serotonin syndrome, an increase in heart rate, and an increase in blood pressure. If you are currently taking any of these medications, please consult with your healthcare provider before using this formulation.

Tetracaine can interact with certain medications as well, including sulfonamides and other local anesthetics. These interactions can increase the risk of side effects such as methemoglobinemia, a serious condition that reduces the amount of oxygen that can be carried in the blood. If you are currently taking any of these medications, please consult with your healthcare provider before using this formulation.

It's also important to note that both Amitriptyline and Tetracaine can interact with certain over-the-counter medications and herbal supplements. For example, taking St. John's Wort with Amitriptyline can increase the risk of serotonin syndrome, while taking Ginkgo Biloba with Tetracaine can increase the risk of bleeding. Please inform your healthcare provider of all medications and supplements you are currently taking to avoid potential interactions.

This formulation is designed to treat specific gynecological conditions such as vulvodynia and vestibulodynia, conditions characterized by chronic vulvar pain without an identifiable cause. The Amitriptyline in the formulation works by changing the way your body feels pain, while the Tetracaine provides immediate relief by numbing the area. This dual-action approach can provide significant relief for women suffering from these conditions.

If you have any questions about this formulation or potential drug interactions, please don't hesitate to reach out to us. We are here to help ensure that you can use this medication safely and effectively.

How Does it Work

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Amitriptyline HCl 1%/Tetracaine HCl 2% Vaginal Cream is a compounded medication that combines two active ingredients, Amitriptyline HCl and Tetracaine HCl, in a cream base. This formulation is designed to be applied directly to the vaginal area to provide localized relief for specific gynecological conditions.

Amitriptyline HCl is a tricyclic antidepressant that has been found to be effective in managing chronic pain. It works by increasing the levels of certain chemicals in the brain that help elevate mood and reduce the sensation of pain. When applied topically in the form of a cream, Amitriptyline HCl can provide targeted pain relief in the area where it is applied. This can be particularly beneficial for conditions such as vulvodynia, a chronic pain condition that affects the vulvar area.

Tetracaine HCl is a local anesthetic that works by blocking nerve signals in your body. When applied to the vaginal area, it can numb the tissue and provide relief from pain or discomfort. This can be particularly beneficial for conditions such as dyspareunia (painful intercourse), or for providing relief during post-surgical recovery.

The cream base of this formulation is designed to be easily applied to the vaginal area. It helps to ensure that the active ingredients are delivered directly to the area where they are needed, providing targeted relief. The cream base also helps to moisturize and soothe the skin, which can be beneficial in managing symptoms such as dryness or irritation.

It's important to note that this is a compounded medication, which means it is made specifically for you, based on a prescription from your healthcare provider. The strength of the active ingredients, as well as the specific combination of ingredients, can be adjusted to best meet your individual needs.

If you have any questions about Amitriptyline HCl 1%/Tetracaine HCl 2% Vaginal Cream, or if you would like more information about how it can be used to manage your specific condition, please don't hesitate to reach out to us. We are here to help and are committed to providing you with the highest level of care.

Other Uses

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Amitriptyline HCl 1%/Tetracaine HCl 2% Vaginal Cream has been formulated primarily to manage specific gynecological conditions. This potent combination can provide relief from genital pain, particularly provoked vestibulodynia, due to Amitriptyline’s properties as a tricyclic antidepressant that can modify the way the body senses pain and Tetracaine’s ability as an anesthetic to temporarily numb the area.

However, this formulation may have other uses beyond its principal indication. It could potentially be applied in other areas demanding localized pain relief or tissue numbing. For example, skin conditions involving neuropathic pain or certain dermatological procedures might benefit from this medication.

The nerve pain medication Amitriptyline can also be employed in treating pain generated from nerves damaged by shingles. In addition, the analgesic Tetracaine can be used in mucosal surfaces of the mouth or throat, to numb the area during dental procedures or swallowing, for instance.

Though it's worth mentioning that off-label use of this formulation demands a doctor’s prescription and supervision. We must underscore the necessity of adhering to the recommended dose and frequency, as misuse can potentially lead to drug resistance, unwanted side effects, or even toxicity.

It’s also critical to inform your doctor about your full medical history, allergies, and other medications taken concurrently, considering that Amitriptyline and Tetracaine can have interactions with other drugs. Be aware that Amitriptyline can cause drowsiness, so let your doctor know if you regularly consume alcohol or take any sedatives.

Undeniably, even though this formulation was made specifically for vaginal application, its components give it real potential for extended use in various other medical domains. We strongly encourage physicians and patients to reach out to us for additional clarifications or information about this formulation. Your safety and satisfaction are our utmost priority.

Frequently Asked Questions

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What is the purpose of the Amitriptyline HCl 1%/Tetracaine HCl 2% Vaginal Cream?

This compounded formulation is designed to deliver medication for specific gynecological conditions in a comfortable, convenient way. It helps deliver therapeutic effects in the vaginal area.

How should this cream be applied?

This semisolid formulation is dispensed in a tube for precise and convenient application in the vaginal area. Please follow your healthcare provider's instructions for usage.

What is the Tetracaine HCl component intended to do?

Tetracaine HCl is a local anesthetic. It works by numbing the skin and surrounding area, which also helps in providing relief from painful conditions.

What is the role of Amitriptyline HCl in this formulation?

Amitriptyline HCl is an antidepressant that also has analgesic properties. It helps in alleviating symptoms associated with certain gynecological conditions when applied topically.

Do I need a prescription to get this cream?

Yes. This cream is a compounded formulation and is not available over-the-counter. It needs to be prescribed by a healthcare provider.

What should I do if I experience any side effects?

If you experience any adverse effects after using this cream, immediately contact your healthcare provider or visit the emergency room.

Can I use this cream while I'm pregnant or breastfeeding?

You should consult with your healthcare provider before using this cream if you are pregnant or breastfeeding, as these conditions may require a different dosing or usage regimen.

Can this cream be used for all gynecological conditions?

No, this cream is intended for specific gynecological conditions and should be used as directed by your healthcare provider.

Can I use this cream if I am having my menstrual period?

You should discuss this with your healthcare provider to get the best advice based on your specific condition and circumstances.

How should I store my Amitriptyline HCl 1%/Tetracaine HCl 2% Vaginal Cream?

Please refer to the manufacturer's guideline for storage. Typically, the cream is stored at room temperature and kept away from heat and direct light. Make sure to keep it out of reach of children.

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Formulas and/or material listed are not to be interpreted as a promise, guarantee or claim of therapeutic efficacy or safety. The information contained herein is not intended to replace or substitute for conventional medical care, or encourage its abandonment. Every patient is unique, and formulas should be adjusted to meet their individual needs.

No compounded medications are reviewed by the FDA for safety or efficacy.