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Compound Catalog

Estradiol Valerate

Estradiol Valerate is a synthetic estrogen used in hormone replacement therapy and various gynecological treatments. It is a prodrug of estradiol, which means it is converted into the active form of estrogen in the body, helping to alleviate symptoms associated with estrogen deficiency.

This API is commonly utilized in formulations designed to manage menopausal symptoms, such as hot flashes and vaginal atrophy, as well as in transgender hormone therapy. Its efficacy in maintaining bone density and cardiovascular health makes it a valuable component in personalized medicine approaches for patients requiring estrogen supplementation.

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Active Ingredient Information

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Estradiol Valerate is a synthetic ester of the naturally occurring estrogen, estradiol, and is commonly used in hormone replacement therapy (HRT) and other hormonal treatments. It is designed to mimic the effects of endogenous estrogen, providing relief from menopausal symptoms such as hot flashes, vaginal dryness, and osteoporosis prevention. By maintaining stable estrogen levels, Estradiol Valerate helps in reducing the risk of cardiovascular diseases and improving overall quality of life for postmenopausal women.

In addition to its use in HRT, Estradiol Valerate is also utilized in transgender hormone therapy, aiding in the development of secondary female sexual characteristics. Its pharmacokinetics involve a gradual release and conversion into estradiol, ensuring a sustained therapeutic effect. This API is often preferred for its predictable absorption and metabolism, which contribute to its efficacy and safety profile. Healthcare providers may consider Estradiol Valerate for patients requiring a tailored approach to estrogen therapy, taking into account individual health needs and treatment goals.

Formulas using

Estradiol Valerate

Formulas and/or material listed are not to be interpreted as a promise, guarantee or claim of therapeutic efficacy or safety. The information contained herein is not intended to replace or substitute for conventional medical care, or encourage its abandonment. Every patient is unique, and formulas should be adjusted to meet their individual needs.

No compounded medications are reviewed by the FDA for safety or efficacy.