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Formulas

Lidocaine 2%/Morphine Sulfate 10 mg/Ketamine HCl 7.5 mg/Diazepam 2.5 mg Suppository

Bayview Pharmacy's Lidocaine 2%/Morphine Sulfate 10 mg/Ketamine HCl 7.5 mg/Diazepam 2.5 mg Suppository is a compounded formulation designed for insertion into a body cavity, typically the rectum or vagina. Upon dissolution or melting, it releases medication for local or systemic absorption. This medication is primarily used for the management of conditions such as chronic pain, neuropathic pain, postoperative pain, fibromyalgia, and migraines.

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Morphine Sulfate
Ketamine Hydrochloride
Diazepam
Lidocaine Hydrochloride
Suppository
6427079ea64324d294518d57
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Formula Information

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This compounded formulation combines Lidocaine 2%, Morphine Sulfate 10 mg, Ketamine HCl 7.5 mg, and Diazepam 2.5 mg into a suppository dosage form. The suppository is a solid dosage form that is inserted into a body cavity, typically the rectum or vagina. Once inserted, it dissolves or melts, releasing the medication for local or systemic absorption.

The formulation is designed to treat a range of conditions including pain, dysmenorrhea, endometriosis, interstitial cystitis, and vulvodynia. Each component of the formulation plays a crucial role in providing relief. Lidocaine and Ketamine HCl are anesthetics that work by blocking nerve signals in the body, thereby providing relief from pain. Morphine sulfate is an opioid analgesic that binds to opioid receptors in the brain, offering relief from moderate to severe pain. Diazepam, a benzodiazepine, increases the activity of the neurotransmitter GABA, providing relief from anxiety and muscle spasms.

This formulation is not only effective in treating the aforementioned conditions, but it also offers additional benefits. It can provide relief from pain, reduce inflammation, and alleviate muscle spasms. Furthermore, it can help reduce anxiety and improve sleep quality.

While this formulation is safe and effective when used as directed, it is crucial to follow your healthcare provider's instructions and take the medication as prescribed. If you have any questions or concerns about this formulation, please do not hesitate to reach out to your healthcare provider or pharmacist for further information and guidance.

Drug Interactions

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This compounded formulation of Lidocaine 2%/Morphine Sulfate 10 mg/Ketamine HCl 7.5 mg/Diazepam 2.5 mg Suppository is a multi-faceted treatment option designed to address a variety of conditions including pain, dysmenorrhea, endometriosis, interstitial cystitis, and vulvodynia. Each component of this formulation plays a crucial role in providing relief.

Lidocaine, a local anesthetic, functions by blocking nerve signals in the area where it's applied, effectively numbing the region and providing pain relief. Morphine sulfate, an opioid analgesic, binds to opioid receptors in the brain and spinal cord, mitigating moderate to severe pain. Ketamine HCl, another anesthetic, operates similarly by blocking nerve signals in the brain and spinal cord, further contributing to pain relief.

Diazepam, a benzodiazepine, enhances the activity of gamma-aminobutyric acid (GABA) in the brain. This action helps to alleviate anxiety and muscle spasms, which can be associated with conditions like endometriosis and interstitial cystitis. Together, these four active ingredients work in synergy to provide comprehensive relief from the symptoms associated with these conditions.

It's crucial to remember that this formulation should only be used under the guidance of a healthcare provider. The suppository is a solid dosage form that is inserted into a body cavity, typically the rectum or vagina, where it dissolves or melts to release the medication for local or systemic absorption. This method of administration allows for targeted treatment, enhancing the efficacy of the medication while minimizing potential side effects.

If you have any questions or concerns about this formulation, it's recommended to consult with your healthcare provider to ensure it's the right treatment option for your specific needs and circumstances.

How Does it Work

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This compounded formulation combines Lidocaine 2%, Morphine Sulfate 10 mg, Ketamine HCl 7.5 mg, and Diazepam 2.5 mg into a suppository form. Each of these components plays a crucial role in managing pain and related conditions. Lidocaine, a local anesthetic, functions by blocking nerve signals in the area where it's applied, thereby providing pain relief. Morphine sulfate, an opioid analgesic, binds to opioid receptors in the brain and spinal cord, offering significant relief from pain. Ketamine HCl, another anesthetic, works similarly by blocking nerve signals in the brain and spinal cord, contributing to pain management. Diazepam, a benzodiazepine, enhances the activity of the neurotransmitter GABA, further aiding in pain relief.

This formulation is designed to be administered rectally as a suppository, where it dissolves or melts to release the medication. This method allows for both local and systemic absorption of the medication, providing targeted and effective relief. It is crucial to follow the instructions provided by your healthcare provider when using this formulation to ensure its efficacy and your safety.

While this formulation is highly effective, it is not intended for prolonged use. It should not be used for more than 7 consecutive days. If you have any questions or concerns about this formulation or its use, it is recommended to consult with your healthcare provider or pharmacist for further guidance.

Other Uses

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This compounded formulation of Lidocaine 2%/Morphine Sulfate 10 mg/Ketamine HCl 7.5 mg/Diazepam 2.5 mg Suppository is a potent treatment option for a variety of pain-related conditions and symptoms. It is particularly effective in managing chronic pain, neuropathic pain, postoperative pain, fibromyalgia, and migraines. Additionally, it can be utilized to alleviate symptoms of muscle spasms, anxiety, and insomnia.

The Lidocaine component of this formulation serves to mitigate pain and inflammation. The Morphine Sulfate is instrumental in reducing pain and relaxing muscles. The Ketamine HCl also contributes to pain reduction and muscle relaxation. The Diazepam component is beneficial in reducing anxiety and promoting sleep.

This formulation can be administered as a single dose or as a continuous treatment, depending on the severity and nature of the condition being treated. It is important for patients to be aware that this formulation may cause side effects such as drowsiness, dizziness, and confusion. As such, it should not be used when operating machinery or driving.

Patients should also be cognizant of the potential for this formulation to interact with other medications. It is strongly recommended that patients consult with their healthcare provider before initiating this treatment. If you have any questions or concerns about this formulation, please do not hesitate to reach out for further information.

Frequently Asked Questions

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What is this compounded formulation of Lidocaine/Morphine Sulfate/Ketamine/Diazepam Suppository?

This is a compounded medication that combines Lidocaine, Morphine Sulfate, Ketamine, and Diazepam into a single suppository. It is a solid dosage form that is inserted into a body cavity, typically the rectum or vagina, where it dissolves or melts to release the medication for local or systemic absorption.

What is the purpose of this compounded formulation?

This compounded formulation is designed to provide pain relief and sedation. The combination of these four medications can provide potent analgesic and sedative effects, which can be beneficial in managing severe pain or anxiety.

How should I use this suppository?

This suppository should be inserted into the rectum or vagina as directed by your healthcare provider. It will dissolve or melt to release the medication. Always wash your hands before and after use.

What are the potential side effects of this compounded formulation?

Side effects can include drowsiness, dizziness, constipation, and dry mouth. More serious side effects can include slow or shallow breathing, severe drowsiness/dizziness, difficulty waking up, or confusion. If you experience any of these side effects, contact your healthcare provider immediately.

Can I use this compounded formulation if I am pregnant or breastfeeding?

Always consult your healthcare provider before using any medication while pregnant or breastfeeding. This compounded formulation may pass into breast milk and may have undesirable effects on a nursing infant.

Can I drive or operate machinery after using this suppository?

This compounded formulation can cause drowsiness or dizziness. Do not drive, use machinery, or do anything that needs alertness until you can do it safely.

What should I do if I miss a dose?

If you miss a dose, use it as soon as you remember. If it is near the time of the next dose, skip the missed dose. Use your next dose at the regular time. Do not double the dose to catch up.

Can I drink alcohol while using this compounded formulation?

Alcohol can increase the risk of serious side effects such as extreme drowsiness/dizziness, slow/shallow breathing, severe drowsiness/dizziness, difficulty waking up. Avoid alcoholic beverages while using this medication.

What should I do in case of an overdose?

If someone has overdosed and has serious symptoms such as passing out or trouble breathing, call emergency services immediately. Symptoms of overdose may include severe drowsiness/dizziness, slow/shallow breathing, severe drowsiness/dizziness, difficulty waking up.

How should I store this compounded formulation?

Store at room temperature away from light and moisture. Do not store in the bathroom. Keep all medications away from children and pets.

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Formulas and/or material listed are not to be interpreted as a promise, guarantee or claim of therapeutic efficacy or safety. The information contained herein is not intended to replace or substitute for conventional medical care, or encourage its abandonment. Every patient is unique, and formulas should be adjusted to meet their individual needs.

No compounded medications are reviewed by the FDA for safety or efficacy.